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Medicinal Chemistry Research Group

Group
Il gruppo di ricerca ha competenze scientifiche nel campo della chimica farmaceutica e della chimica organica di sintesi; possiede un’esperienza consolidata nella progettazione, sintesi e valutazione biologica di peptidi modificati o peptidomimetici inibitori di proteasi quali efficaci agenti terapeutici per il trattamento di patologie tumorali o di patologie causate da protozoi e da virus.
Address:
Viale F. Stagno d'Alcontres, 31 - 98166 Messina
date/time interval:
(October 2, 2000 - )
  • Overview
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Overview

Term type

Altro gruppo di ricerca

Linked Units

Dipartimento di Scienze chimiche, biologiche, farmaceutiche e ambientali

Research Fields

Concepts (4)


PE5_18 - Medicinal chemistry - (2020)

Goal 3: Good health and well-being

Settore CHIM/08 - Chimica Farmaceutica

Settore CHEM-07/A - Chimica farmaceutica

Keywords (4)

  • ascendant
  • decrescent
Drug design
Inibitori di proteasi
Peptidomimetici
Sintesi peptidica
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Overview

Design, synthesis and biological evaluation of peptidomimetics as inhibitors of human, viral, protozoan proteases
No Results Found

Affiliation

Has member (2)

ETTARI Roberta
ZAPPALA' Maria

List of all contributors

Collaborazione con gruppi di ricerca esterni, Prof. Sandro Cosconati Dipartimento di Scienze e Tecnologie Ambientali Biologiche e Farmaceutiche Università della Campania Luigi Vanvitelli., Prof. Tanja Schirmeister Institute of Pharmacy and Biochemistry University of Mainz DE., Prof. Conor Caffrey Skaggs School of Pharmacy and Pharmaceutical Sciences University of California San Diego (USA)., Prof. Philip Rosenthal Department of Medicine at the University of California San Francisco (USA)., Prof. Lorenzo Corsi Dipartimento di Scienze della Vita Università di Modena e Reggio Emilia, Dr. Florine Cavelier Institut des Biomolécules Max Mousseron Univerity of Montpellier FR., Prof. Michael Gutschow Pharmaceutical Institute - Pharmaceutical & Medicinal Chemistry University of Bonn DE., Prof. Steven Ballet Organic Chemistry Research Group Vrije Universiteit Brussel BE., Dr. Clément Morgat Department of Nuclear Medicine & Radiopharmacy University of Bordeaux FR., Prof. John Ziebuhr Institute of Medical Virology Justus Liebig University Giessen DE., Prof. Graciela Andrei Molecular Structural and Translational Virology Research Group University of Leuven BE.

Members (5)

CALABRO' Maria
DI CHIO Carla
PREVITI Santo
STARVAGGI JOSÈ
TOTARO NOEMI

Contact

Email address (2)

rettari@unime.it
mzappala@unime.it

Equipments & Resources

Equipments

Spettrometro NMR Varian 500
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